99% Ukucoceka kwePeptide Hormone BreMelanotide PT 141 CAS 189691-06-3
Iinkcukacha ngokukhawuleza:
Igama lemveliso
|
PT-141 |
Izibizo |
I-Brmelanotice, iBreMelanotide Acetate, iBremelanotide |
CAS Hayi |
Ngo-189691-06-3 |
MF |
C50H69N15O10 |
MW |
1040.17736 |
Ucoceko |
99% |
Inkangeleko |
Umgubo omhlophe |
IBakala |
KwiBanga lezeMayeza |
Iphuhlisiwe ukusuka kwiMelanotan II
I-Bremelanotide okanye i-PT-141, ikhemikhali yophando kunye ne-peptide, yeyokuhlelwa okubizwa ngokuba yi-melanocyte evuselela iihormone (MSH). Yi-hexapeptide analog ye-alpha-MSH, kwaye yaveliswa kwasekuqaleni isuka kwi-MSH Melanotan II, iarhente ye-peptide eyaphononongwa kwizilingo zokutshiswa ngaphandle kwelanga kodwa, ngequbuliso, kukhokelele ekuvuseleleni ngokwesondo kunye nokuzimela okuzenzekelayo ngokwesondo kwizifundo ezilithoba zovavanyo ezilishumi.
I-Bremelanotide yikhompawundi ephantsi kwesiyobisi njengonyango lokungasebenzi kakuhle kwabasetyhini nabesilisa, ukothuka okwenzakalisayo kunye nokulimala okuphinda kwenzeke.
Unyango lokungasebenzi kakuhle ngokwesondo
I-Bremelanotide okanye i-PT-141 ligama eliqhelekileyo le-peptide entsha yophando yokusetyenziswa ekuncedeni ukuphucula ukungasebenzi ngokwesondo emadodeni (ukungasebenzi kakuhle kwe-erectile okanye ukungabi namandla) kunye nokunceda ukuphucula ukungasebenzi kakuhle ngokwesondo kwabasetyhini (ukuphazamiseka kwesini).
I-PT-141 sisixhobo esinokubakho kunyango lokungasebenzi kakuhle ngokwesondo; ngakumbi ukungasebenzi kakuhle kwamadoda. I-Bremelanotide, i-PT-141 ayisebenzi kwinkqubo ye-vascular efana nezinto zangaphambili kodwa iyaziwa kwaye ibonakalisiwe ukunceda ukwandisa isenzo sezesondo kwizilwanyana ezanyisayo ezingamadoda nabasetyhini. I-Bremelanotide PT-141 kuthiwa isebenza ngokwenza i-melanocortin receptors kwingqondo, ke oko kunceda ukonyusa ukonyusa isondo.
I-Bremelanotide lunyango lwenoveli olunokuthi lubutshintshe ubuso bokunyanga ukuphazamiseka kwezesondo, hayi kuphela ngenxa yokusebenza kwayo ngenxa yendlela eyahlukileyo yokwenza, kodwa nangenxa yokhuseleko lwayo kunye nenyani yokuba isebenza ngokudibeneyo nolunye unyango lwe-ED / SAD.
I-Bremelanotide iyasebenza kumandla ayo okunyanga ukuphazamiseka kweminqweno yesini kunye nokuphazamiseka okuchaphazela ukuvuswa komzimba. I-Bremelanotide inyusa i-Lordosis kwizifundo zezilwanyana, umqondiso wokuzilungiselela ngokwasemzimbeni wokukhuphela. Kwamadoda, ayikhuthazi imeko ye-vascular yelungu lobudoda, kodwa endaweni yoko isebenza ukuvuselela inkqubo ye-nervous system ikakhulu ngokusebenzisa umsebenzi we-dopamine receptor ukunyusa umnqweno wesini kwaye ikwabonisa ukusebenza kunyango olusebenzayo lwe-ED / SAD, ngokunokwenzeka ngokuphucula umqondiso .
Ukulawulwa ngokudibeneyo kwe-PT-141 kunye neSildenafil
I-Bremelanotide ikwabonelela ngokubakho njengonyango oluphantsi lwedosi ephantsi kunye ne-sildenafil yedosi esezantsi. Impendulo ye-erectile ebangelwa kukulawulwa ngokubambisana kwe-PT-141 kunye ne-sildenafil yayinkulu kakhulu kunempendulo eyayibangelwa kukulawulwa kwe-sildenafil yodwa. Ukulawulwa ngokudibeneyo kwe-PT-141 kunye ne-sildenafil yayikhuselekile kwaye inyamezelwe kakuhle kwaye ayikhange ibangele izehlo ezimbi okanye iziganeko ezichaseneyo ezonyuswe rhoqo okanye ubungqongqo xa kuthelekiswa ne-monotherapy. Isithinteli sinokwenza enye indlela yokunyanga kwizigulana ekungenazo idosi ephezulu yonyango olunye ezinganyamezelekiyo okanye ezinganyamezelekiyo.
Uncedo:
1. Amava atyebileyo. Sele sikhethekile kule nkalo kangangeminyaka, sinamava atyebileyo kunye nenethiwekhi yentengiso ebanzi ejikeleze igama. I-steroid yethu kunye neehomoni zithunyelwe kumazwe aphesheya, njengeYurophu, iAfrika, iAsia, iMelika kunye namanye amazwe. Asinayo ingxelo elungileyo evela kwindwendwe lethu, kodwa sisekwe ubudlelwane beshishini olude kunye nabo.
2. Umgangatho omkhulu kunye nococeko oluphezulu. Umgangatho omnye yimfihlo yempumelelo yethu. Zonke iimveliso zethu zinandipha ukucoceka okuphezulu. Ke, inokuqinisekisa ukuba iimfuno zabaxhasi bethu. Wamkelekile umyalelo weesampulu, i-MOQ iigram ezili-10 kuphela.
3. Ukuhanjiswa okukhuselekileyo kunye okukhawulezayo. Sinesitokhwe sobunzima, ukuze sikwazi ukwenza amalungiselelo okuhanjiswa ngaphakathi kweeyure ezingama-24 sakuba sifumene intlawulo. Inombolo yokulandelela iya kwaziswa ngokukhawuleza emva kokuthunyelwa. Sinendlela yethu yokupakisha enokuthi ithumele i-0.01 yeekhilo ukuya kwiimveliso ezingama-50 zeekhilogram ngexesha.
4. Inkonzo elungileyo yasemva kokuthengisa. 24/7 iyafumaneka. Siza kukuxelela ulwazi oluhlaziyiweyo lwephakheji ye-ASAP. Kwaye zama konke okusemandleni ethu ukusombulula iingxaki ezahlukeneyo abahlangabezana nazo abathengi
5. Ukuthenga okunamava. Ngaphandle kwepowder eluhlaza eluhlaza kunye nolwelo, sinika isisombululo sehomoni kunye nefomula. Sinokukufundisa ngendlela yokwenza isisombululo sehomoni kwindawo leyo. Naluphi na utyelelo kwilebhu yethu lwamkelekile
Ezinye iiMveliso
Ioksijini |
50-56-6 |
98.0% imiz |
Ipamorelin |
Ngo-170851-70-4 |
99.07% |
ISermorelin Acetate |
Ngama-86168-78-7 |
98.0% imiz |
IHGH 176-191 |
|
Iipesenti ezingama-98 |
BPC 157 |
137525-51-0 |
99% |
MT-2 |
121062-08-6 |
Iipesenti ezingama-98 |
GHRP-6 |
87616-84-0 |
98.0% imiz |
GHRP-2 |
158861-67-7 |
98.0% imiz |
PT-141 |
Ngo-189691-06-3 |
99% |
Epithalon |
307297-39-8 |
99% |
FST344 |
Ngo-189691-06-3 |
99% |